Dihexa (PNB-0408)

Peptide

Dihexa (N-hexanoic-Tyr-Ile-(6) aminohexanoic amide) is an angiotensin IV-derived peptide that potentiates hepatocyte growth factor (HGF)/c-Met receptor signaling. Preclinical studies show remarkable cognitive enhancement at picomolar concentrations. In Alzheimer's disease mouse models, dihexa restored cognitive function and promoted synaptogenesis. Seven orders of magnitude more potent than BDNF in promoting dendritic spine formation. Currently investigational with no completed human clinical trials.

Quick Answer

What it is

Dihexa (N-hexanoic-Tyr-Ile-(6) aminohexanoic amide) is an angiotensin IV-derived peptide that potentiates hepatocyte growth factor (HGF)/c-Met receptor signaling. Preclinical studies show remarkable cognitive enhancement at picomolar concentrations.

Key findings

  • Grade C: Cognitive Enhancement (Cognitive Function)
  • Grade C: Synaptogenesis (Cognitive Function)
  • Grade C: Neuroprotection (Cognitive Function)

Safety

No specific caution or interaction language was detected in the current summary/outcome notes.

⚠️ Research Notice

This peptide information is for educational and research purposes only. Peptides may not be FDA-approved for human use and may only be legally available for research purposes. Consult qualified healthcare professionals before considering any peptide compounds.

ℹ️ Quick Facts: Dihexa (PNB-0408)

Quick Facts: Dihexa (PNB-0408)

  • Best Evidence:Grade C
  • Conditions Studied:1
  • Research Outcomes:5
  • Key Effect:Cognitive Function
A0
B0
C4
D1
1 conditions · 5 outcomes

Detailed Outcomes

C
Cognitive Enhancement
Preclinical: Restored spatial learning and memory in aged rats and APP/PS1 Alzheimer's mice. 7 orders of magnitude more potent than BDNF for spinogenesis. Reversed scopolamine-induced deficits. No human trial data available.
largeImproves
C
Synaptogenesis
Preclinical: Promoted new dendritic spine formation in hippocampal neurons at picomolar concentrations. Enhanced synaptic connectivity and plasticity via HGF/c-Met/PI3K pathway activation.
largeImproves
C
Neuroprotection
Preclinical: Protected against neurodegeneration in Alzheimer's mouse models. Reduced amyloid-related cognitive decline. Enhanced neuronal survival via c-Met signaling.
moderateImproves
D
Lipid Profile
2 preclinical studies support this finding. Primarily preclinical evidence.
smallImproves

Research Citations (15)

Efficiently generate functional hepatic cells from human pluripotent stem cells by complete small-molecule strategy.
(2022)
PMID: 35410439
Dihexa Improves Cognitive Deficits in Aged Rats by Promoting Hippocampal Synaptogenesis
(2021)
PMID: 34827486
Cognitive benefits of angiotensin IV and angiotensin-(1-7): A systematic review of experimental studies.
(2018)
PMID: 29733881
Hepatocyte Growth Factor/c-Met Signaling in Head and Neck Cancer and Implications for Treatment
(2017)
PMID: 30455415
Brain angiotensin system in cognitive function: involvement of AT4 receptors
(2017)
PMID: 29122679
Small-Molecule-Directed Hepatocyte-Like Cell Differentiation of Human Pluripotent Stem Cells.
(2016)
PMID: 27532814
The angiotensin AT4 receptor subtype as a target for the treatment of memory dysfunction associated with Alzheimer's disease
(2015)
PMID: 25649658
Hepatocyte growth factor mimetic protects lateral line hair cells from aminoglycoside exposure.
(2015)
PMID: 25674052
Small-molecule-driven hepatocyte differentiation of human pluripotent stem cells.
(2015)
PMID: 25937370
Effect of structure on the interactions between five natural antimicrobial compounds and phospholipids of bacterial cell membrane on model monolayers.
(2014)
PMID: 24914896

Related Peptides

Tesamorelin

Peptide

1 shared condition · 15 outcomes

Tesamorelin is a 44-amino-acid synthetic analog of growth hormone-releasing hormone (GHRH) that is FDA-approved (2010) for reducing excess abdominal fat in HIV-infected patients with lipodystrophy. It stimulates endogenous pulsatile GH secretion from the pituitary gland. Tesamorelin has demonstrated efficacy in reducing visceral adipose tissue, liver fat (NAFLD), and improving cognitive function in clinical trials.

Sermorelin

Peptide

1 shared condition · 18 outcomes

Sermorelin (GHRH 1-29) is a 29-amino-acid synthetic analog of growth hormone-releasing hormone (GHRH) that retains full biological activity. It was FDA-approved in 1990 for diagnostic use and in 1997 for treating childhood growth hormone deficiency. Sermorelin stimulates natural GH release from the pituitary gland through the hypothalamic-pituitary axis, producing physiological GH patterns with built-in safety through somatostatin feedback regulation.

Semax

Peptide

1 shared condition · 14 outcomes

Semax is a synthetic heptapeptide derived from ACTH (adrenocorticotropic hormone). It has been approved as a prescription medication in Russia and Ukraine for treating stroke, cognitive disorders, and peptic ulcers. Research suggests it may enhance BDNF expression and exhibit nootropic and neuroprotective effects. Most clinical research has been conducted in Russia, with limited Western clinical trials.

Selank

Peptide

1 shared condition · 9 outcomes

Selank is a synthetic heptapeptide derived from tuftsin, an immunomodulatory peptide. It has been approved in Russia as a treatment for anxiety and neurasthenic conditions. Research indicates it may have anxiolytic, nootropic, and immunomodulatory properties without sedative effects. Like Semax, most clinical research has been conducted in Russia.

Pinealon

Peptide

1 shared condition · 4 outcomes

Pinealon is a synthetic tripeptide (Glu-Asp-Arg) developed by Russian researchers as part of the Khavinson peptide bioregulators. It is designed to target brain tissue and has been studied for potential neuroprotective and cognitive-enhancing effects. Research suggests it may help regulate circadian rhythms and support cognitive function in aging, though human clinical data is limited.